Amidepsine A

SKU
A-1430
  • Formula:C29H29NO11
  • MW:567.6
  • Appearance:White to Pale Yellow Powder
  • Purity:95% (HPLC)
Product Name Qty
Amidepsine A
1 mg
$276.96
Amidepsine A
2.5 mg
$519.29

Inhibitor of diacylglycerol acyltransferase (DGAT). Shows inhibitory effect in rat liver microsomes (IC=10.2 M) and Raji cells (IC=15.5 M). Excessive accumulation of triacetylglycerol produced by DGAT may cause fatty liver, obesity and hypertriglyceridemia, which may lead to atherosclerosis, diabetes and metabolic disorders.

More Information
SKU
A-1430
Chemical Name
2,4-DIMETHOXY-6-METHYL-BENZOIC ACID 4-[[4-[[(1-CARBOXYETHYL)AMINO]CARBONYL]-3-HYDROXY-5-METHYLPHENOXY]CARBONYL]-3-HYDROXY-5-METHYLPHENYL ESTER
Chemical Formula
C29H29NO11
Molecular Weight
567.6
Appearance
White to Pale Yellow Powder
Purity
95% (HPLC)
Solubility
Soluble in methanol or ethyl acetate; insoluble in water.
Stability
N/A
Storage Temp
-20°C
THERAPEUTIC AREA
Vascular Disorders
USE
Amidepsine A is an inhibitor of DGAT (diacylglycerol acyltransferase) use in atherosclerosis, diabetes and metabolic disorders
MDL NUMBER
MFCD28138425
CHEMACX
Not Applicable
INCHI
InChI=1S/C29H29NO11/c1-13-8-18(10-20(31)23(13)26(33)30-16(4)27(34)35)40-28(36)24-14(2)9-19(11-21(24)32)41-29(37)25-15(3)7-17(38-5)12-22(25)39-6/h7-12,16,31-32H,1-6H3,(H,30,33)(H,34,35)
SMILES
CC1=CC(=CC(=C1C(=O)NC(C)C(=O)O)O)OC(=O)C2=C(C=C(C=C2C)OC(=O)C3=C(C=C(C=C3C)OC)OC)O
Peptide sequence
Not Applicable
RTECS
Not Applicable
UN #'S
Not Applicable
PACKING GROUP
Not Applicable
HAZARD CLASS
Not Applicable
Promo text for AGS discount
N/A
GHS PICTOGRAMS
UN #'S Not Applicable
Packing Group Not Applicable
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