Derquantel

SKU
D-2499
  • CAS:187865-22-1
  • Formula:C28H37N3O4
  • MW:479.6
  • Appearance:White solid
  • Purity:>98% by HPLC
Product Name Qty
Derquantel
25 mg
$1,196.02
Derquantel
5 mg
$341.72
*Please inquire the availability for this product. Derquantel is a semi-synthetic paraherquamide analogue prepared by removal of the 2-oxo group in a four-step sequence of N-protection, reduction, N-deprotection and a final reduction. Derquantel is a potent nematocide and was the first paraherquamide to be successfully commercialised in combination with avermectin. Derquantel, like other paraherquamides, induces a flaccid paralysis in nematodes thought to be due to inhibition of nicotinic acetylcholine receptors acting as an antagonist of acetylcholine.
More Information
Alternate Name/Synonyms
2-Deoxoparaherquamide, 2-Deoxoparaherquamide A, 2-Desoxoparaherquamide A, PF 00520904, PNU 141962
SKU
D-2499
CAS #
187865-22-1
Chemical Formula
C28H37N3O4
Molecular Weight
479.6
Appearance
White solid
Purity
>98% by HPLC
Solubility
Soluble in ethanol, methanol, DMSO, DMF, and water (poorly)
Storage Temp
-20°C
MDL NUMBER
MFCD13195549
INCHI
InChI=1S/C28H37N3O4/c1-23(2)10-12-34-21-18(35-23)8-7-17-20(21)29-15-26(17)14-27-16-31-11-9-25(5,33)28(31,22(32)30(27)6)13-19(27)24(26,3)4/h7-8,10,12,19,29,33H,9,11,13-16H2,1-6H3/t19-,25+,26-,27+,28-/m0/s1
SMILES
C[C@]1(CCN2[C@]13C[C@@H]4[C@](C2)(C[C@]5(C4(C)C)CNc6c5ccc7c6OC=CC(O7)(C)C)N(C3=O)C)O
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