EPZ6438

SKU
E-2511
  • CAS:1403254-99-8
  • Formula:C34H44N4O4
  • MW:572.74
  • Appearance:white powder
  • Purity:≥99%
Product Name Qty
EPZ6438
25 mg
$222.16
EPZ6438
100 mg
$673.20
EPZ6438
1 mg
$44.88
EPZ6438
5 mg
$84.15

EPZ-6438 is an inhibitor of EZH2, a histone methyltransferase (HMT) responsible for methylation of lysine and arginine residues and controls gene transcription fidelity in cells. EPZ-6438 displays anticancer chemotherapeutic activity in in vivo models by inducing regression of malignant or atypical teratoid rhabdoid tumors containing altered or mutant SWI/SNF ATP-dependent chromatin remodelers.

More Information
Alternate Name/Synonyms
E7438, Tazemetostat
SKU
E-2511
CAS #
1403254-99-8
Chemical Name
N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-[ethyl(oxan-4-yl)amino]-2-methyl-5-[4-(morpholin-4-ylmethyl)phenyl]benzamide
Chemical Formula
C34H44N4O4
Molecular Weight
572.74
Appearance
white powder
Purity
≥99%
Solubility
In DMSO
Storage Temp
-20°C
Hazard Image
Yes
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