GW501516

SKU
G-2348
  • CAS:317318-70-0
  • Formula:C21H18F3NO3S2
  • MW:453.5
  • Appearance:White to off-white Solid
  • Purity:98% by HPLC

0

0

0

0

Product Name Qty
GW501516
1 mg
$165.17
GW501516
5 mg
$615.10

A selective agonist for PPAR (peroxisome proliferator-activated receptor) (EC= 1. 1 nM), displaying 1000-fold selectivity over the other human subtypes. In macrophages, fibroblasts, and intestinal cells, GW501516 increases expression of the reverse cholesterol transporter ATP-binding cassette A1 and induces apolipoprotein A1-specific cholesterol efflux.

More Information
Alternate Name/Synonyms
(2-Methyl-4-(((4-methyl-2-(4-trifluoromethylphenyl)-1,3-thiazol-5-yl)methyl)sulfanyl)phenoxy)acetic acid
SKU
G-2348
CAS #
317318-70-0
Chemical Name
(2-Methyl-4-(((4-methyl-2-(4-trifluoromethylphenyl)-1,3-thiazol-5-yl)methyl)sulfanyl)phenoxy)acetic acid
Chemical Formula
C21H18F3NO3S2
Molecular Weight
453.5
Appearance
White to off-white Solid
Purity
98% by HPLC
Solubility
DMSO (50 mg/ml) or EtOH (12 mg/ml)
Stability
N/A
Storage Temp
-20°C
THERAPEUTIC AREA
Endocrinological Disorders
USE
A selective and potent PPARβ agonist
MDL NUMBER
MFCD09033000
CHEMACX
X1463059-2
PubChecm ID
N/A
INCHI
InChI=1S/C21H18F3NO3S2/c1-12-9-16(7-8-17(12)28-10-19(26)27)29-11-18-13(2)25-20(30-18)14-3-5-15(6-4-14)21(22,23)24/h3-9H,10-11H2,1-2H3,(H,26,27)
SMILES
CC1=C(C=CC(=C1)SCC2=C(N=C(S2)C3=CC=C(C=C3)C(F)(F)F)C)OCC(=O)O
Peptide sequence
Not Applicable
RTECS
AI9105500
UN #'S
Not Applicable
PACKING GROUP
Not Applicable
HAZARD CLASS
Not Applicable
Handling
Protect from light and air
Special Shipping
N/A
E-Guides
N/A
Blog Post
N/A
Citations
N/A
Citations_Hyperlink
N/A
Reference
N/A
Reference Hyperlink
N/A
Additional Images
N/A
Additional Videos
N/A
Hazard Image
N/A
Promo text for AGS discount
N/A
Handling Protect from light and air
UN #'S Not Applicable
Packing Group Not Applicable
To Top