Kenpaullone

SKU

K-1050

CAS:142273-20-9
Formula:C₁₆H₁₁BrN₂O
MW:327.2
Appearance:Tan/Brown Powder
Purity:>95%

SDS

CofA

Product Name	Qty
Kenpaullone 1 mg $55.81
Kenpaullone 5 mg $227.82

Details

Paullones represent a novel class of small molecule cyclin-dependent kinase (CDK) inhibitors. Kenpaullone is a potent inhibitor of CDK1/cyclin B (IC₅₀=400 nM) also inhibits CDK2/cyclin A (IC₅₀=680 nM). Weaker effect on other kinases. Also shown to inhibit GSK-3β (IC₅₀=23 nM)

Specifications

More Information

SKU

K-1050

CAS #

142273-20-9

Chemical Name

9-Bromo-7,12-dihydroindolo-[3,2-d][1]benzazepin-6(5H)-one

Chemical Formula

C₁₆H₁₁BrN₂O

Molecular Weight

327.2