SDS
CofA
Paullones represent a novel class of small molecule cyclin-dependent kinase (CDK) inhibitors. Kenpaullone is a potent inhibitor of CDK1/cyclin B (IC50=400 nM) also inhibits CDK2/cyclin A (IC50=680 nM). Weaker effect on other kinases. Also shown to inhibit GSK-3β (IC50=23 nM)
More Information
SKU
K-1050
CAS #
142273-20-9
Chemical Name
9-Bromo-7,12-dihydroindolo-[3,2-d][1]benzazepin-6(5H)-one
Chemical Formula
C16H11BrN2O
Molecular Weight
327.2
Appearance
Tan/Brown Powder
Purity
>95%
Solubility
Soluble in DMSO (>25mg/ml). Insoluble in Water, or Ethanol.
Storage Temp
-20°C
Certificate of Analysis 1
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