PPAR-gamma Antagonist, G3335

SKU
P-2406
  • CAS:36099-95-3
  • Formula:C16H19N3O5
  • MW:333.34
  • Appearance:White Solid
  • Purity:97% by elemental analysis
Product Name Qty
PPAR-gamma Antagonist, G3335
10 mg
$75.94
PPAR-gamma Antagonist, G3335
25 mg
$150.77
Cell-permeable. A dipeptide that acts as a selective and reversible PPARg antagonist (KD ~ 8 M). Shown to inhibit the agonist activity of Rosiglitazone (100 nM) in a dose-dependent manner (IC= 31.9 M) in transfected COS-7 cells.
More Information
Alternate Name/Synonyms
G3335; H-Trp-Glu-OH
SKU
P-2406
CAS #
36099-95-3
Chemical Name
2-[[2-AMINO-3-(1H-INDOL-3-YL)PROPANOYL]AMINO]PENTANEDIOIC ACID
Chemical Formula
C16H19N3O5
Molecular Weight
333.34
Appearance
White Solid
Purity
97% by elemental analysis
Solubility
Soluble in Water
Stability
N/A
Storage Temp
-20°C
THERAPEUTIC AREA
Endocrinological Disorders
USE
A cell-permeable dipeptide that acts as a selective PPAR-γ antagonist used in diabetes
MDL NUMBER
MFCD00037964
CHEMACX
X1096243-7
INCHI
InChI=1S/C16H19N3O5/c17-11(7-9-8-18-12-4-2-1-3-10(9)12)15(22)19-13(16(23)24)5-6-14(20)21/h1-4,8,11,13,18H,5-7,17H2,(H,19,22)(H,20,21)(H,23,24)/t11-,13-/m0/s1
SMILES
C1=CC=C2C(=C1)C(=CN2)C[C@@H](C(=O)N[C@@H](CCC(=O)O)C(=O)O)N
Peptide sequence
Not Applicable
RTECS
Not Applicable
UN #'S
Not Applicable
PACKING GROUP
Not Applicable
HAZARD CLASS
Not Applicable
Handling
Protect from light and mositure
Certificate of Analysis 1
Promo text for AGS discount
N/A
Handling Protect from light and mositure
UN #'S Not Applicable
Packing Group Not Applicable
To Top