DMSO (50 mg/ml) or EtOH (12 mg/ml)
A selective agonist for PPAR (peroxisome proliferator-activated receptor) (EC= 1. 1 nM), displaying 1000-fold selectivity over the other human subtypes. In macrophages, fibroblasts, and intestinal cells, GW501516 increases expression of the reverse cholesterol transporter ATP-binding cassette A1 and induces apolipoprotein A1-specific cholesterol efflux.
Research or further manufacturing use only, not for food or drug use.