328968-36-1
445.4
C24H19N3O6
DMF, DMSO
-20°C
Cell-permeable. A reversible, p300/CBP (CREB-binding protein) histone acetyltransferase (HAT) inhibitor (K = 400 nM). Specific inhibition to p300 (86%) compared to N-acetyltransferase, PCAF, GCN5, Rtt109, Sas or MOZ histone acetyltransferases (10%). Suppresses histone H3 and H4 acetylation in mouse fibroblast cell lines.
0.1 lbs
Research or further manufacturing use only, not for food or drug use.