388082-78-8
925.46
C29H26ClFN4O4S.2C7H8O3S
DMSO (200 mg/ml)
-20°C
Lapatinib is a potent inhibitor of EGFR kinase (K = 3 nM), ErbB-2 kinase (K = 13 nM), ErbB-4 kinase (K = 347 nM). Lapatinib can restore tamoxifen sensitivity in tamoxifen-resistant, ER-positive breast cancer models.
0.1 lbs
Research or further manufacturing use only, not for food or drug use.