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Price$ 343.72
  • SKU: B-2201-5MG
  • Pack Size: 5 MG
Quantity
-
+

501437-28-1

391.42

C19H23F2N5O2

Soluble in DMSO (>25 mg/ml)

-20°C


Cell-permeable. ATP-competitive inhibitor of the four isoforms of ribosomal S6 kinase (p90 RSK) (IC's at 100 M ATP: RSK1 = 31 nM, RSK2 = 24 nM, RSK3 = 18 nM, RSK4 = 15 nM). Does not significantly inhibit 10 other AGC kinases, and over 40 other protein kinases at 100X concentrations. In addition, BI-D1870 completely prevents PMA-induced TSC2 (a regulator of mTORC1) phosphorylation at Ser.

0.1 lbs



Research or further manufacturing use only, not for food or drug use.

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