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Celastrol, 100 MG

Price$ 863.99
  • SKU: C-2262-100MG
  • Pack Size: 100 MG





Methanol: Clear red solution at 10 mg/mL



Celastrol (also known as Tripterin) is a cell-permeable proteasome inhibitor. Acts as an antioxidant, anti-inflammatory and immunosuppressive agent. Suppresses LPS-induced cytokine release in macrophages and monocytes (IC= 40 nM for IL-1 and IL-1, 80 nM for IL-6, 110 nM for prostaglandin E2 and 210 nM for IL-8 and TNF). Suppresses nitric oxide (NO) production (IC= 230 nM) and LPS-induced NF-B activation (IC= 270 nM).Inhibits chymotrypsin-like activity of 20S proteasome (IC= 2.5 M) and lipid peroxidation induced by ADP and Fe in rat liver mitochondria (IC= 7 M).

Isolated from Tripterygium wilfordii.


0.1 lbs

Research or further manufacturing use only, not for food or drug use.

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