- Appearance:White to off-white Solid
- Purity:98% by HPLC
Cell-permeable. A potent inhibitor of the human epidermal growth factor receptor 2 (HER2) tyrosine kinase (IC= 6 nM). Displays > 4000-fold selectivity over EGFR, FGFR, PDGFR, JAK1 and Src. TAK 165 inhibits bladder, kidney and androgen-independent prostate cancer in vitro and in vivo.
|Handling||Protect from light and air|
|UN #'S||Not Applicable|
|Packing Group||Not Applicable|