TGX-221
SKU
T-2460
- CAS:663619-89-4
- Formula:C21H24N4O2
- MW:364.44
- Appearance:White Solid
- Purity:98% by HPLC


Cell-permeable. A potent, selective and ATP-competitive inhibitor of PI 3-kinase (IC= 5 nM for p110). Inhibits other PI3K isoforms at higher concentrations (IC= 0.1 M for p110, 5 M for p110, and 3.5 M for p110).
More Information
Alternate Name/Synonyms
7-Methyl-2-(morpholin-4-yl)-9-(1-phenylaminoethyl)-pyrido[1,2-a]-pyrimidin-4-one
SKU
T-2460
CAS #
663619-89-4
Chemical Name
(±)-7-Methyl-2-(morpholin-4-yl)-9-(1-phenylaminoethyl)-pyrido[1,2-a]-pyrimidin-4-one
Chemical Formula
C21H24N4O2
Molecular Weight
364.44
Appearance
White Solid
Purity
98% by HPLC
Solubility
DMSO (10 mg/ml) or Ethanol (5 mg/ml)
Storage Temp
-20°C
THERAPEUTIC AREA
Not Available
USE
Not Available
MDL NUMBER
MFCD11113209
CHEMACX
X1600331-3
INCHI
InChI=1S/C21H24N4O2/c1-15-12-18(16(2)22-17-6-4-3-5-7-17)21-23-19(13-20(26)25(21)14-15)24-8-10-27-11-9-24/h3-7,12-14,16,22H,8-11H2,1-2H3
SMILES
CC1=CN2C(=O)C=C(N=C2C(=C1)C(C)NC3=CC=CC=C3)N4CCOCC4
Peptide sequence
Not Applicable
RTECS
Not Applicable
UN #'S
Not Applicable
PACKING GROUP
Not Applicable
HAZARD CLASS
Not Applicable
Handling
Protect from air and light
Handling | Protect from air and light |
---|---|
UN #'S | Not Applicable |
Packing Group | Not Applicable |