Zaprinast

SKU
Z-1001
  • CAS:37762-06-4
  • Formula:C13H13N5O2
  • MW:271.3 Da
  • Appearance:White solid
  • Purity:>98% by HPLC

0

0

0

Product Name Qty
Zaprinast
100 mg
$212.19
Zaprinast
20 mg
$52.48

Description

Zaprinast is a cell-permeable, selective inhibitor of cGMP-specific phosphodiesterase (PDE V) (IC₅₀ = 0.45 µM). Inhibits PDE IX only at higher concentrations (IC₅₀ = 35 µM).

More Information
Alternate Name/Synonyms
Zaprinastum; 2-o-Propoxyphenyl-8-azapurine-6-one
SKU
Z-1001
CAS #
37762-06-4
Chemical Name
5-(2-propoxyphenyl)-2,6-dihydrotriazolo[4,5-d]pyrimidin-7-one
Chemical Formula
C13H13N5O2
Molecular Weight
271.3 Da
Appearance
White solid
Purity
>98% by HPLC
Solubility
Soluble inDMSO (25mg/mL), or 100% ethanol (5 mg/mL). Insoluble in water.
Melting Point
N/A
Preparation
N/A
Storage Temp
Room temperature
THERAPEUTIC AREA
N/A
USE
A cell-permeable, selective inhibitor of cGMP-specific phosphodiesterase.
Merck Index
N/A
MDL NUMBER
MFCD00214073
CHEMACX
X1065780-2
INCHI
InChI=1S/C13H13N5O2/c1-2-7-20-9-6-4-3-5-8(9)11-14-12-10(13(19)15-11)16-18-17-12/h3-6H,2,7H2,1H3,(H2,14,15,16,17,18,19)
SMILES
CCCOC1=CC=CC=C1C2=NC(=O)C3=NNNC3=N2
Peptide sequence
N/A
RTECS
XZ6157358
UN #'S
N/A
PACKING GROUP
N/A
HAZARD CLASS
N/A
Handling
Further processing of solid materials may result in the formation of combustible dusts. The potential for combustible dust formation should be taken into consideration before additional processing occurs. Provide appropriate exhaust ventilation at places where dust is formed.
Certificate of Analysis 1
GHS PICTOGRAMS
Handling Further processing of solid materials may result in the formation of combustible dusts. The potential for combustible dust formation should be taken into consideration before additional processing occurs. Provide appropriate exhaust ventilation at places where dust is formed.
To Top